Keynote Talk VI
Structure-Based Design in Drug Discovery and Process Chemistry
Recommended Reading:
A Real-World Perspective on Molecular Design
Bernd Kuhn et al.
J. Med. Chem., 2016, 59 (9), pp 4087–4102
Systematic Approach to Conformational Sampling for Assigning Absolute Configuration Using Vibrational Circular Dichroism
Edward C. Sherer et al.
J. Med. Chem., 2014, 57, pp 477–494
Interrogating Selectivity in Catalysis using Molecular Vibrations
Anat Milo, Elizabeth N. Bess & Matthew S. Sigman
Nature 2014, 507, 210–214
Modeling a Crowdsourced Definition of Molecular Complexity
Robert P. Sheridan et al.
J. Chem. Inf. Model., 2014, 54 (6), pp 1604–1616
A Multifunctional Catalyst that Stereoselectively Assembles Prodrugs
Daniel A. DiRocco*, Yining Ji, Edward C. Sherer, Artis Klapars, Mikhail Reibarkh, James Dropinski, Rose Mathew, Peter Maligres, Alan M. Hyde, John Limanto, Andrew Brunskill, Rebecca T. Ruck, Louis-Charles Campeau, Ian W. Davies
Science 2017, 356, 426-430
DOI: 10.1126/science.aam7936